APS03118 [Ligand Id: 14205] activity data from GtoPdb

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  • ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949]
GtoPdb Potency for RET V804M - 9.9 pIC50 0.13 nM IC50 J Med Chem (2025) : [PMID:40920215]
GtoPdb Potenct for WT RET - 10.02 pIC50 0.09 nM IC50 J Med Chem (2025) : [PMID:40920215]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.