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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885] | ||||||||
GtoPdb | Binding affinity for BRD4 BD2 | - | 8 | pKd | <10 | nM | Kd | US20220204500A1. Compounds comprising n-methyl-2-pyridone, and pharmaceutically acceptable salts (2025) |
GtoPdb | Binding affinity for BRD4 BD1 | - | 8 | pKd | <10 | nM | Kd | US20220204500A1. Compounds comprising n-methyl-2-pyridone, and pharmaceutically acceptable salts (2025) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.